Exelixis Drug Patent Portfolio

Exelixis owns 1 orange book drug protected by 7 US patents Given below is the list of Exelixis's drug patents along with their expiration dates.

Drug Patent Number Drug Patent Title Drug Patent Expiry Status
US11298349 Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds 10 Feb, 2032
Active
US9717720 Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds 10 Feb, 2032
Active
US8877776 (L)-malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide 08 Oct, 2030
Active
US11091439 Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N′-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms therof for the treatment of cancer 15 Jan, 2030
Active
US11091440 Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)- N′-(4-fluorophenyl)cyclopropane-1,1 -dicarboxamide, and crystalline forms thereof for the treatment of cancer 15 Jan, 2030
Active
US11098015 Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N′-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancer 15 Jan, 2030
Active
US7579473 c-Met modulators and methods of use 14 Aug, 2026
Active


Given below is the list of recent legal activities going on the following drug patents of Exelixis.

Activity Date Patent Number
Patent litigations
Payment of Maintenance Fee, 8th Year, Large Entity 20 Apr, 2022 US8877776
Recordation of Patent Grant Mailed 12 Apr, 2022 US11298349
Patent Issue Date Used in PTA Calculation 12 Apr, 2022 US11298349
Email Notification 24 Mar, 2022 US11298349
Issue Notification Mailed 23 Mar, 2022 US11298349
Application Is Considered Ready for Issue 18 Mar, 2022 US11298349
Dispatch to FDC 18 Mar, 2022 US11298349
Email Notification 10 Mar, 2022 US11298349
Mail Response to 312 Amendment (PTO-271) 10 Mar, 2022 US11298349
Response to Amendment under Rule 312 04 Mar, 2022 US11298349
Pubs Case Remand to TC 01 Mar, 2022 US11298349
Email Notification 28 Feb, 2022 US11298349
Mail PUB other miscellaneous communication to applicant 28 Feb, 2022 US11298349
Amendment after Notice of Allowance (Rule 312) 28 Feb, 2022 US11298349
PUB Other miscellaneous communication to applicant 24 Feb, 2022 US11298349


Exelixis Drug Patents' Oppositions Filed in EPO

Exelixis drug patents have faced multiple oppositions in the European Patent Office. The earliest opposition was filed on Dec 05, 2013, by Actavis Group Ptc Ehf. This opposition was filed on patent number EP10701175A. Click below to reveal the latest opposition data.


Application Filing Date Opposition Party Legal Status
Patent litigations
EP12704492A Aug, 2022 STADA Arzneimittel AG Revoked
EP10701175A Dec, 2013 Ladendorf, Oliver Patent maintained as amended
EP10701175A Dec, 2013 Gallafent, Alison Patent maintained as amended
EP10701175A Dec, 2013 Actavis Group PTC ehf Patent maintained as amended


Exelixis's Family Patents

Exelixis drugs have patent protection in a total of 31 countries. It's US patent count contributes only to 23.9% of its total global patent coverage. 1 country has all of their patents expired or invalidated which has opened up potential generic launch opportunities in this particular country. Click below to unlock the full patent family tree.

Family Patents



Exelixis Drug List

Given below is the complete list of Exelixis's drugs and the patents protecting them.


1. Cometriq

Cometriq is protected by 7 patents, out of which none have expired yet. Check out its patent list below.

Drug Patent Number Drug Patent Title Drug Patent Expiry Status
US11298349 Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds 10 Feb, 2032
(7 years from now)
Active
US9717720 Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds 10 Feb, 2032
(7 years from now)
Active
US8877776 (L)-malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide 08 Oct, 2030
(5 years from now)
Active
US11091439 Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N′-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms therof for the treatment of cancer 15 Jan, 2030
(5 years from now)
Active
US11091440 Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)- N′-(4-fluorophenyl)cyclopropane-1,1 -dicarboxamide, and crystalline forms thereof for the treatment of cancer 15 Jan, 2030
(5 years from now)
Active
US11098015 Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N′-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancer 15 Jan, 2030
(5 years from now)
Active
US7579473 c-Met modulators and methods of use 14 Aug, 2026
(1 year, 8 months from now)
Active

Discover which of these patents contain the active ingredient(API) of the drug, their family patents, along with litigation and legal activity details of these patents on Cometriq's drug page


Explore Our Curated Drug Screens

Drugs Generating Over $1 Billion in Annual Revenue
Explore the top-performing drugs that dominate the pharmaceutical industry
View List
NCE-1 Patent Expiry in the Next 1 Year
Identify opportunities as new chemical entity (NCE-1) patents approach expiry
View List
Recently Granted Patents in EP
Find the opportunity to file Oppositions
View List