Rare Lung Diseases Therapeutics

1. Rapamune patent expiration

Treatment: Inhibiting transplant rejection using rapamycin (sirolimus)

Drug Patent Number Company Drug Patent Title Drug Patent Expiry Activity Alert
These drug patents focus on the other aspects of the active substance like dosage, mode of administration (oral, tablet, capsules, liquids etc).
US5536729 PF PRISM CV Rapamycin formulations for oral administration
Sep, 2013

(12 years ago)

US5100899 PF PRISM CV Methods of inhibiting transplant rejection in mammals using rapamycin and derivatives and prodrugs thereof
Jul, 2013

(12 years ago)

US5989591 PF PRISM CV Rapamycin formulations for oral administration
Mar, 2018

(7 years ago)

US5536729

(Pediatric)

PF PRISM CV Rapamycin formulations for oral administration
Mar, 2014

(11 years ago)

US5100899

(Pediatric)

PF PRISM CV Methods of inhibiting transplant rejection in mammals using rapamycin and derivatives and prodrugs thereof
Jan, 2014

(12 years ago)

US5403833

(Pediatric)

PF PRISM CV Methods of inhibiting transplant rejecton in mammals using rapamycin and derivatives and prodrugs thereof
Oct, 2012

(13 years ago)

US5989591

(Pediatric)

PF PRISM CV Rapamycin formulations for oral administration
Sep, 2018

(7 years ago)




Drug Exclusivity Drug Exclusivity Expiration
Orphan Drug Exclusivity(ODE) May 28, 2022
Orphan Drug Exclusivity(ODE-92) May 28, 2022

Drugs and Companies using SIROLIMUS ingredient

Market Authorisation Date: 15 September, 1999

Dosage: SOLUTION; TABLET

How can I launch a generic of RAPAMUNE before it's drug patent expiration?
More Information on Dosage

RAPAMUNE family patents

Family Patents