Lumateperone Tosylate Patent Expiration

Lumateperone Tosylate is Used for treating schizophrenia, bipolar depression, and bipolar disorder by modulating serotonin and dopamine receptor activity. It was first introduced by Intra-Cellular Therapies Inc in its drug Caplyta on Dec 20, 2019.


Lumateperone Tosylate Patents

Given below is the list of patents protecting Lumateperone Tosylate, along with the drug name that holds that patent and the company name owning that drug.

Drug Used in Drug Patent Number Drug Patent Title Drug Patent Expiry Drug Owner
Caplyta US11753419 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)phenyl)butan-1-one for treating conditions of the central nervous system and cardiac disorders Dec 10, 2040 Intra-cellular
Caplyta US12122792 Pharmaceutical compositions comprising 4-((6bR,10aS)-3-methyl2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin8(7H)-yl)-1-(4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)phenyl)butan-1-one for treating conditions of the central nervous system and cardiac disorders Dec 10, 2040 Intra-cellular
Caplyta US12090155 Methods Jul 07, 2040 Intra-cellular
Caplyta US11980617 Methods of treating acute depression and/or acute anxiety Oct 27, 2039 Intra-cellular
Caplyta US10695345 Pharmaceutical capsule compositions comprising lumateperone mono-tosylate Aug 30, 2039 Intra-cellular
Caplyta US11052084 Pharmaceutical capsule compositions comprising lumateperone mono-tosylate Aug 30, 2039 Intra-cellular
Caplyta US11690842 Pharmaceutical capsule compositions comprising lumateperone mono-tosylate Aug 30, 2039 Intra-cellular
Caplyta US11806348 Methods of treatment using pharmaceutical capsule compositions comprising lumateperone mono-tosylate Aug 30, 2039 Intra-cellular
Caplyta US12070459 Pharmaceutical capsule compositions comprising lumateperone mono-tosylate Aug 30, 2039 Intra-cellular
Caplyta US12128043 Pharmaceutical capsules comprising lumateperone mono-tosylate Aug 30, 2039 Intra-cellular
Caplyta US10960009 Methods of treating schizophrenia and depression Dec 03, 2034 Intra-cellular
Caplyta US11026951 Methods of treating bipolar disorder Dec 03, 2034 Intra-cellular
Caplyta US9956227 Method for the treatment of residual symptoms of schizophrenia Dec 03, 2034 Intra-cellular
Caplyta USRE48839 Methods and compositions for sleep disorders and other disorders Aug 19, 2033 Intra-cellular
Caplyta US8598119 Methods and compositions for sleep disorders and other disorders Dec 28, 2029 Intra-cellular
Caplyta US8648077 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone toluenesulfonic acid addition salt and salt crystals Dec 01, 2029 Intra-cellular
Caplyta US10117867 Methods and compositions for sleep disorders and other disorders May 27, 2029 Intra-cellular
Caplyta US9168258 Methods and compositions for sleep disorders and other disorders May 27, 2029 Intra-cellular
Caplyta US9616061 Methods and compositions for sleep disorders and other disorders May 27, 2029 Intra-cellular
Caplyta US9199995 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone toluenesulfonic acid addition salt and salt crystals Mar 12, 2029 Intra-cellular
Caplyta US9586960 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de] quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone toluenesulfonic acid salt crystal forms Mar 12, 2029 Intra-cellular
Caplyta USRE48825 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone toluenesulfonic acid salt crystal forms Mar 12, 2029 Intra-cellular
Caplyta USRE48825 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone toluenesulfonic acid salt crystal forms Feb 12, 2029 Intra-cellular
Caplyta US10464938 Pharmaceutical compositions comprising ((6bR,10aS)-1-(4-fluorophenyl)-4-(3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)butan-1-one or pharmaceutically acceptable salts thereof Mar 12, 2028 Intra-cellular
Caplyta US7183282 Substituted heterocycle fused γ-carbolines Jun 15, 2020

(Expired)

Intra-cellular
Caplyta USRE39680 Substituted heterocycle fused gamma-carbolines Jun 15, 2020

(Expired)

Intra-cellular



Lumateperone Tosylate's Family Patents

Family Patents

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