Bosutinib Monohydrate Patent Expiration

Bosutinib Monohydrate is used for treating BCR-ABL positive leukemia resistant to imatinib, including patients with specific BCR-ABL mutations and various phases of CML. It was first introduced by Pf Prism Cv in its drug Bosulif on Sep 4, 2012.


Bosutinib Monohydrate Patents

Given below is the list of patents protecting Bosutinib Monohydrate, along with the drug name that holds that patent and the company name owning that drug.

Drug Used in Drug Patent Number Drug Patent Title Drug Patent Expiry Drug Owner
Bosulif US11103497 Treatment of imatinib resistant leukemia Feb 28, 2034 Pf Prism Cv
Bosulif US11103497

(Pediatric)

Treatment of imatinib resistant leukemia Aug 28, 2034 Pf Prism Cv
Bosulif US6002008 Substituted 3-cyano quinolines Mar 27, 2018

(Expired)

Pf Prism Cv
Bosulif US6002008 Substituted 3-cyano quinolines Mar 27, 2018

(Expired)

Pf Prism Cv
Bosulif US7417148 4-anilino-3-quinolinecarbonitriles for the treatment of chronic myelogenous leukemia (CML) Dec 11, 2025 Pf Prism Cv
Bosulif US7417148

(Pediatric)

4-anilino-3-quinolinecarbonitriles for the treatment of chronic myelogenous leukemia (CML) Jun 11, 2026 Pf Prism Cv
Bosulif US7767678 Crystalline forms of 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methyl-1-piperazinyl)propoxy]-3-quinolinecarbonitrile and methods of preparing the same Nov 23, 2026 Pf Prism Cv
Bosulif US7767678

(Pediatric)

Crystalline forms of 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methyl-1-piperazinyl)propoxy]-3-quinolinecarbonitrile and methods of preparing the same May 23, 2027 Pf Prism Cv
Bosulif US7919625 4-anilino-3-quinolinecarbonitriles for the treatment of chronic myelogenous leukemia (CML) Dec 11, 2025 Pf Prism Cv
Bosulif US7919625

(Pediatric)

4-anilino-3-quinolinecarbonitriles for the treatment of chronic myelogenous leukemia (CML) Jun 11, 2026 Pf Prism Cv
Bosulif USRE42376 Substituted 3-cyanoquinolines Apr 13, 2024

(Expired)

Pf Prism Cv
Bosulif USRE42376

(Pediatric)

Substituted 3-cyanoquinolines Oct 13, 2024 Pf Prism Cv


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